SCHEMBL8617024

SCHEMBL8617024

COC(=O)c1cc(-c2ccccc2)nc2c(OC)cccc12

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.81
DHODH Q02127 2/20 0.61
PLA2G2A P14555 5/20 0.60
ALDH1A1 P00352 3/20 0.57
HPGD P15428 3/20 0.57
CCR6 P51684 1/20 0.57
ACACA Q13085 2/20 0.55
KDM4E B2RXH2 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
MAPT P10636 4/20 0.53
TP53 P04637 2/20 0.53
POLB P06746 1/20 0.52
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616292 0.90 PDE10A (1.00) PDE10ADHODHALDH1A1HPGDCCR6
SCHEMBL8617709 0.83 PDE10A (0.69) PDE10ADHODHALDH1A1HPGDCCR6
SCHEMBL2576382 0.81 KDM4E (0.76) PDE10ADHODHPLA2G2AALDH1A1HPGD
SCHEMBL30690053 0.81 PLA2G2A (0.73) PDE10ADHODHPLA2G2AALDH1A1HPGD
SCHEMBL6659920 0.80 TACR3 (0.74) PDE10AALDH1A1KDM4EMEN1KMT2A
SCHEMBL8617941 0.79 PDE10A (0.64) PDE10ADHODHALDH1A1HPGDACACA
SCHEMBL11395164 0.78 PDE10A (0.67) PDE10AALDH1A1HPGDACACAKDM4E
SCHEMBL3902043 0.78 DHODH (0.62) PDE10ADHODHPLA2G2AALDH1A1HPGD
SCHEMBL7826492 0.77 PDE10A (0.77) PDE10ADHODHALDH1A1HPGDCCR6
SCHEMBL8876443 0.77 PDE10A (0.52) PDE10ADHODHPLA2G2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed