SCHEMBL8617709

SCHEMBL8617709

COc1cccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc12

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.69
ACACA Q13085 2/20 0.54
ALDH1A1 P00352 5/20 0.48
HPGD P15428 2/20 0.48
CYP3A4 P08684 1/20 0.47
DHODH Q02127 2/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
MAPT P10636 5/20 0.46
KDM4E B2RXH2 5/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
POLB P06746 1/20 0.46
ALOX12 P18054 1/20 0.46
HTT P42858 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
GAA P10253 1/20 0.45
CCR6 P51684 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617941 0.96 PDE10A (0.64) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8615321 0.89 PDE10A (0.54) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8615313 0.89 PDE10A (0.54) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8620680 0.89 ALDH1A1 (0.54) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8614875 0.87 PDE10A (0.52) PDE10AALDH1A1HPGDCYP3A4DHODH
SCHEMBL8616298 0.87 PDE10A (0.52) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8613395 0.86 PDE10A (0.51) PDE10AACACAALDH1A1HPGDCYP3A4
SCHEMBL8614344 0.86 PDE10A (0.52) PDE10AACACAALDH1A1HPGDDHODH
SCHEMBL8615931 0.85 PDE10A (0.51) PDE10AACACAALDH1A1CYP3A4MEN1
SCHEMBL8615930 0.85 PDE10A (0.51) PDE10AACACAALDH1A1CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed