SCHEMBL8617520

SCHEMBL8617520

O=C(NCSc1ccncc1)c1cccnc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.63
NPC1 O15118 3/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
ALDH1A1 P00352 2/20 0.63
THRB P10828 1/20 0.60
ROCK2 O75116 1/20 0.55
ROCK1 Q13464 1/20 0.55
KMT2A Q03164 6/20 0.55
MEN1 O00255 5/20 0.55
GAA P10253 1/20 0.54
HDAC1 Q13547 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
TSHR P16473 1/20 0.51
ALOX15 P16050 1/20 0.51
HSD17B10 Q99714 1/20 0.51
EPHX2 P34913 2/20 0.50
MAPT P10636 1/20 0.50
CYP1A2 P05177 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966814 0.83 RAB9A (0.72) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL29572289 0.80 THRB (0.66) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL14415899 0.77 THRB (0.77) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL25328235 0.77 THRB (0.77) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL19028142 0.77 TSHR (0.76) RAB9ANPC1SMN1; SMN2THRBROCK2
N-Hydroxymethylnicotinamide SCHEMBL352358 0.76 THRB (1.00) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL1233991 0.74 THRB (0.72) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL17822214 0.74 EPHX2 (0.75) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL9786935 0.74 THRB (0.72) RAB9ANPC1SMN1; SMN2ALDH1A1THRB
SCHEMBL31314589 0.74 THRB (0.72) RAB9ANPC1SMN1; SMN2ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767121-A ANTIINFLAMMATORY AND -ARTHRITIC AGENTS; ANTIPYRETICS; ANALGESICS; ADHESION PROTEIN EXPRESSION AND CYCLOXYGENASE AND 5-LIPOXYGENASE INHIBITORS; IMMUNOSUPPRESSANTS AND -MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-16 US disclosed
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
EP-0522606-B1 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-04-03 EP disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed