SCHEMBL8617898

SCHEMBL8617898

C=C(c1ccc(N)cc1)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.48
MAOB P27338 3/20 0.48
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 2/20 0.44
HTT P42858 1/20 0.44
GFER P55789 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
LMNA P02545 3/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
PRMT1 Q99873 1/20 0.41
TSHR P16473 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALOX15 P16050 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41
MASP2 O00187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL725856 0.87 MAPT (0.55) MAOAMEN1KMT2AMAPTHTT
SCHEMBL1796583 0.87 MAPT (0.55) MAOAMAOBMAPTHTTGFER
4-Chloroaniline SCHEMBL27544 0.79
4-Chloroaniline SCHEMBL16922177 0.79
SCHEMBL10905142 0.78 CA1 (0.42) MAOAMAOBMEN1KMT2AMAPT
SCHEMBL9823021 0.78 MEN1 (0.54) MAOAMAOBMEN1KMT2AMAPT
SCHEMBL3695975 0.78 CES2 (0.60) MAOAMAOBMEN1KMT2AMAPT
SCHEMBL4747566 0.76 SRD5A2 (0.64) MAOAMAOBMEN1KMT2AMAPT
SCHEMBL18661442 0.76 ACHE (0.62) MAOAMEN1KMT2AMAPTHTT
SCHEMBL6465868 0.76 MAPT (0.44) MAOAMAOBMAPTHTTGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632017-B1 N-phenyl-2-cyano-3-hydroxy propenamides, their tautomeres and salts, their use as medicaments and compositions containing them HOECHST MARION ROUSSEL INC (FR) 1998-05-06 EP disclosed
US-5416112-A Antiinflammatory agents ROUSSEL UCLAF (FR) 1995-05-16 US disclosed
EP-0632017-A1 N-phenyl-2-cyano-3-hydroxy propenamides, their tautomeres and salts, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1995-01-04 EP disclosed
US-4587361-A N-(4-(1-PHENYLETHENYL)PHENYL)-2-HYDROXY-3,5-DIHALOBENZAMIDE SMITHKLINE BECKMAN CORPORATION (US) 1986-05-06 US disclosed