SCHEMBL8618352

SCHEMBL8618352

CC(C)(C)ON(C=O)C(C=CCOCc1ccccc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.40
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PPARG P37231 1/20 0.36
ALOX5 P09917 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
SLC1A1 P43005 3/20 0.34
SLC1A3 P43003 2/20 0.34
SLC1A2 P43004 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
TK1 P04183 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619514 0.76
SCHEMBL6401312 0.73 CA1 (0.40) PPARAHTTNPSR1PPARGL3MBTL1
SCHEMBL7646162 0.73 PPARA (0.39) PPARANPSR1PPARGL3MBTL1CTSB
SCHEMBL28233244 0.72 CYP1A2 (0.41) PPARAPPARGMAPTCYP1A2
SCHEMBL8618349 0.71 PPARA (0.60) PPARAPPARGCTSBCTSS
SCHEMBL8618354 0.71 PPARA (0.60) PPARAPPARGCTSBCTSS
SCHEMBL8621499 0.70 SLC1A1 (0.49) ALOX5MAPTSLC1A1SLC1A3SLC1A2
SCHEMBL8026778 0.70 L3MBTL1 (0.35) PPARAMAPTL3MBTL1SLC1A1SLC1A3
SCHEMBL20583924 0.70 FOLH1 (0.41) L3MBTL1MEN1KMT2A
SCHEMBL6305685 0.70 FOLH1 (0.41) L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710324-A AMINE CONTAINING COMPOUNDS MERRELL PHARMACEUTICALS INC. (US) 1998-01-20 US disclosed
US-5318992-A Administering for the treatment of hypotensive conditions and shock MERRELL DOW PHARMACEUTICALS INC. (US) 1994-06-07 US disclosed
EP-0446699-A1 Inhibitors of nitric oxide biosynthesis MERRELL PHARMACEUTICALS INC. (US) 1991-09-18 EP disclosed