Biguanide

Biguanide

SCHEMBL8618876

CC(C)(C)c1cc(C(=O)O)cc(C(=O)O)c1.N=C(N)NC(=N)N

nearest known ligand 0.45

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 4/20 0.45
RXRB P28702 4/20 0.45
RXRG P48443 1/20 0.45
DHODH Q02127 1/20 0.44
TDP1 Q9NUW8 2/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
BLM P54132 1/20 0.41
CASP7 P55210 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SRD5A2 P31213 1/20 0.41
CYP1A2 P05177 1/20 0.40
NR1H4 Q96RI1 3/20 0.39
EPHX2 P34913 2/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166878 0.83 RXRB (0.59) RXRARXRBRXRGDHODHTDP1
SCHEMBL14534692 0.82 DHODH (0.60) RXRARXRBRXRGDHODHTDP1
Hydrochloric Acid SCHEMBL11879619 0.81 RXRB (0.57) RXRARXRBRXRGDHODHTDP1
Hydrochloric Acid SCHEMBL4585979 0.81 RXRB (0.57) RXRARXRBRXRGDHODHTDP1
Water SCHEMBL28383353 0.81 RXRB (0.57) RXRARXRBRXRGDHODHTDP1
SCHEMBL8168277 0.81 HDAC3 (0.46) RXRARXRBRXRGTDP1TP53
Hydrochloric Acid SCHEMBL8505491 0.79 HDAC3 (0.45) RXRARXRBRXRGTDP1TP53
SCHEMBL501957 0.79 RXRB (0.64) RXRARXRBRXRGDHODHTDP1
SCHEMBL6362506 0.78 RXRA (0.50) RXRARXRBRXRGDHODHTDP1
SCHEMBL5873298 0.77 RXRB (0.62) RXRARXRBRXRGDHODHTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US claimed
JP-9169718-A None JP disclosed
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
JP-H09169718-A SUBSTITUTED BENZENEDICARBOXYLIC ACID DIGUANIDIDE, ITS PRODUCTION, USE OF THE SAME COMPOUND AS MEDICINE OR DIAGNOSING AGENT AND MEDICINE CONTAINING THE SAME HOECHST AG 1997-06-30 JP disclosed