SCHEMBL8618914

SCHEMBL8618914

Cc1cc(Cl)cc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.46
PPARA Q07869 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 2/20 0.44
ALOX12 P18054 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
RXFP1 Q9HBX9 2/20 0.44
PTGER4 P35408 2/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
KCNH2 Q12809 1/20 0.43
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8619359 0.99 CYP2C9 (0.46) CYP2C9PPARAMEN1KMT2AALDH1A1
SCHEMBL8613481 0.85 KDM4E (0.56) CYP2C9MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8619775 0.82 PPARA (0.64) CYP2C9PPARAMEN1KMT2AALDH1A1
SCHEMBL8617805 0.82 CA12 (0.59) CYP2C9MEN1KMT2AALDH1A1CYP3A4
SCHEMBL8613361 0.82 KDM4E (0.52) CYP2C9MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8618761 0.81 MEN1 (0.56) CYP2C9PPARAMEN1KMT2AALDH1A1
SCHEMBL8614035 0.80 CA12 (0.59) CYP2C9MEN1KMT2AALDH1A1CA12
SCHEMBL8617908 0.79 MEN1 (0.55) CYP2C9PPARAMEN1KMT2AALDH1A1
SCHEMBL8613185 0.79 PDE10A (0.49) CYP2C9MEN1KMT2AALDH1A1CYP2C19
SCHEMBL8619386 0.79 LMNA (0.52) CYP2C9MEN1KMT2AALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed