SCHEMBL8618939

SCHEMBL8618939

Cc1cc(C)cc(-c2cc(NC(=N)NC=O)c3ccccc3n2)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 4/20 0.44
PDE10A Q9Y233 2/20 0.44
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
CYP3A4 P08684 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
MOK Q9UQ07 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618948 0.91 MEN1 (0.50) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8615355 0.91 PDE10A (0.55) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8617753 0.89 ACP1 (0.51) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8618203 0.87 HTT (0.40) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8618150 0.86 KDM4E (0.48) ACP1PDE10AKMT2AMEN1HTT
SCHEMBL8615248 0.86 ACP1 (0.44) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8615676 0.85 ACP1 (0.48) ACP1ABCB1ABCG2CYP3A4
SCHEMBL8617739 0.85 ALDH1A1 (0.47) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8620932 0.85 POLB (0.51) ACP1PDE10AABCB1ABCC1ABCG2
SCHEMBL8614345 0.84 ABCG2 (0.44) ACP1ABCB1ABCC1ABCG2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed