SCHEMBL8618946

SCHEMBL8618946

CC(C)CCCc1ccc(-c2cc(C(=O)NC(=N)N)c3ccccc3n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.56
TSHR P16473 1/20 0.52
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
HPGD P15428 1/20 0.50
THRB P10828 1/20 0.50
LMNA P02545 3/20 0.49
RECQL P46063 1/20 0.49
TACR3 P29371 3/20 0.49
TP53 P04637 3/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MITF O75030 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617937 0.87 PLA2G2A (0.58) DHODHKDM4EALDH1A1MAPTNPC1
SCHEMBL8616548 0.85 TACR3 (0.52) DHODHKDM4EALDH1A1SMN1; SMN2LMNA
SCHEMBL8615123 0.84 DHODH (0.59) DHODHTSHRKDM4EALDH1A1MAPT
SCHEMBL8619733 0.83 DHODH (0.58) DHODHTSHRKDM4EALDH1A1NPC1
SCHEMBL8617743 0.82 CYP3A4 (0.65) DHODHKDM4EALDH1A1SMN1; SMN2MEN1
SCHEMBL8615443 0.82 ALDH1A1 (0.42) DHODHTSHRALDH1A1TACR3CYP2C9
SCHEMBL8614837 0.82 TACR3 (0.60) DHODHKDM4EALDH1A1MAPTNPC1
SCHEMBL8615354 0.81 CYP3A4 (0.65) KDM4EALDH1A1MAPTSMN1; SMN2MEN1
SCHEMBL8619034 0.81 DHODH (0.57) DHODHKDM4EALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL8620745 0.81 CYP3A4 (0.64) DHODHKDM4EALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed