SCHEMBL8619210

SCHEMBL8619210

N=C(NC=O)Nc1cc(-c2cccc(C3CC3)c2)nc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
ACP1 P24666 11/20 0.40
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618001 0.95 DHODH (0.46) ABCB1ABCC1ABCG2ACP1DHODH
SCHEMBL8617753 0.86 ACP1 (0.51) ABCB1ABCC1ABCG2ACP1
SCHEMBL8617828 0.85 DHODH (0.45) ABCB1ABCC1ABCG2ACP1DHODH
SCHEMBL8619887 0.84 DHODH (0.47) ABCB1ABCC1ABCG2ACP1DHODH
SCHEMBL8614861 0.84 AKR1C3 (0.53) ABCB1ABCC1ABCG2ACP1
SCHEMBL8614778 0.83 ACP1 (0.43) ABCB1ABCC1ABCG2ACP1DHODH
SCHEMBL8614345 0.83 ABCG2 (0.44) ABCB1ABCC1ABCG2ACP1
SCHEMBL8614079 0.83 ACP1 (0.52) ABCB1ABCC1ABCG2ACP1
SCHEMBL8615255 0.83 ABCG2 (0.53) ABCB1ABCC1ABCG2ACP1
SCHEMBL8618948 0.83 MEN1 (0.50) ABCB1ABCC1ABCG2ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed