SCHEMBL8617828

SCHEMBL8617828

N=C(NC=O)Nc1cc(-c2ccccc2)nc2cc(C3CCCC3)ccc12

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.45
ACP1 P24666 3/20 0.40
TACR3 P29371 1/20 0.38
ADORA1 P30542 7/20 0.38
ADORA2A P29274 5/20 0.38
ADORA3 P0DMS8 3/20 0.38
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619887 0.99 DHODH (0.47) DHODHACP1TACR3ADORA1ADORA2A
SCHEMBL8618001 0.88 DHODH (0.46) DHODHACP1ABCB1ABCC1ABCG2
SCHEMBL8619210 0.85 ABCB1 (0.41) DHODHACP1ABCB1ABCC1ABCG2
SCHEMBL8617753 0.83 ACP1 (0.51) ACP1ABCB1ABCC1ABCG2
SCHEMBL8615210 0.82 TACR3 (0.44) ACP1TACR3ABCB1ABCC1ABCG2
SCHEMBL8620212 0.81 SGK1 (0.38) ACP1TACR3ADORA1ADORA2AADORA3
SCHEMBL8615938 0.81 TACR3 (0.41) ACP1TACR3ABCB1ABCC1ABCG2
SCHEMBL8619389 0.81 TACR3 (0.41) DHODHACP1TACR3ADORA3ABCB1
SCHEMBL8618234 0.81 RXFP1 (0.44) ACP1TACR3ABCB1ABCC1ABCG2
SCHEMBL8617739 0.81 ALDH1A1 (0.47) ACP1TACR3ABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed