Biguanide

Biguanide

SCHEMBL8619381

N=C(N)NC(=N)N.O=C(O)c1cc(C(=O)O)cc(-c2ccc(Cl)cc2Cl)c1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.54
ALPL P05186 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
CRHBP P24387 1/20 0.44
RAB9A P51151 1/20 0.44
CRHR2 Q13324 1/20 0.44
MARS1 P56192 3/20 0.44
AHR P35869 1/20 0.42
SRD5A1 P18405 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
PYGL P06737 1/20 0.39
SHMT1 P34896 1/20 0.38
SHMT2 P34897 1/20 0.38
DHODH Q02127 1/20 0.38
BCL2L1 Q07817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779218 0.87 SRD5A2 (0.68) SRD5A2ALPLSMN1; SMN2KDM4ENPC1
Biguanide SCHEMBL8614462 0.79 TPMT (0.52) DHODH
Biguanide SCHEMBL8617033 0.77 KMO (0.45) NPC1RAB9ACASP1DHODH
SCHEMBL444367 0.74 SRD5A2 (0.90) SRD5A2SMN1; SMN2KDM4ENPC1CRHBP
SCHEMBL442436 0.73 SRD5A2 (0.62) SRD5A2NPC1RAB9AMARS1SHMT1
SCHEMBL358511 0.70 SRD5A2 (0.48) SRD5A2ALPLSMN1; SMN2KDM4ENPC1
Isophthalic Acid SCHEMBL27991768 0.70 CA1 (0.50) TSHR
SCHEMBL2408930 0.69 CA1 (0.56) SRD5A2SMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL2908235 0.69 NOTUM (0.66) SRD5A2ALPLSMN1; SMN2MARS1AHR
SCHEMBL30069186 0.69 NOTUM (0.66) SRD5A2ALPLSMN1; SMN2MARS1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US claimed
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed