Biguanide

Biguanide

SCHEMBL8617033

N=C(N)NC(=N)N.O=C(O)c1cc(C(=O)O)cc(-c2ccc(F)c(Cl)c2)c1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.45
CASP1 P29466 1/20 0.44
RPA1 P27694 1/20 0.44
DHODH Q02127 4/20 0.43
ICMT O60725 1/20 0.43
ERCC1 P07992 1/20 0.41
ERCC4 Q92889 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
RXRA P19793 2/20 0.40
RXRB P28702 2/20 0.40
ACLY P53396 2/20 0.40
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
ABL1 P00519 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779130 0.87 KMO (0.55) KMOCASP1RPA1DHODHICMT
Biguanide SCHEMBL8614462 0.81 TPMT (0.52) KMODHODHRXRARXRB
Biguanide SCHEMBL8619381 0.77 SRD5A2 (0.54) CASP1DHODHNPC1RAB9A
SCHEMBL3643412 0.76 RXRA (0.61) KMORPA1ERCC1ERCC4RXRA
Hydrochloric Acid SCHEMBL8505392 0.73 KCNQ3 (0.48) NPC1RAB9A
SCHEMBL8297932 0.71 MAP4K4 (0.54) KMOCASP1RPA1ICMTERCC1
Isophthalic Acid SCHEMBL27991768 0.69 CA1 (0.50) KMO
SCHEMBL30308290 0.69 TSHR (0.65) KMORPA1NPC1RAB9ARXRA
SCHEMBL109599 0.69 TSHR (0.65) KMORPA1NPC1RAB9ARXRA
SCHEMBL16608990 0.68 RPA1 (0.58) KMOCASP1RPA1DHODHERCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US claimed
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed