SCHEMBL8620846

SCHEMBL8620846

CC(C)(C)OC(=O)NC[CH]Cc1ccc(O)c(O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.42
KDM4E B2RXH2 4/20 0.41
MAPT P10636 4/20 0.41
HPGD P15428 4/20 0.41
HSD17B10 Q99714 4/20 0.41
ALDH1A1 P00352 3/20 0.41
LMNA P02545 3/20 0.41
BLM P54132 3/20 0.41
HIF1A Q16665 2/20 0.41
PTGS1 P23219 1/20 0.41
POLB P06746 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
ALOX15 P16050 2/20 0.41
THPO P40225 2/20 0.41
ALOX12 P18054 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
XDH P47989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749285 0.81 ERCC1 (0.56) HDAC1GAAERCC1ERCC4CA1
SCHEMBL4583679 0.80 IDO1 (0.53) IDO1CA1NAMPTKDM4A
SCHEMBL30423117 0.79 MAPT (0.63) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL233765 0.79 MAPT (0.63) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL23086057 0.75 ALOX15 (0.46) HDAC1KDM4EMAPTHPGDHSD17B10
SCHEMBL7517472 0.74 MEN1 (0.58) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL2404127 0.74 TDP1 (0.50) KDM4ELMNATDP1GAAMEN1
SCHEMBL27575347 0.72 TDP1 (0.46) KDM4EMAPTTDP1GAAMEN1
SCHEMBL8620843 0.72 ALOX15 (0.50) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL8790742 0.72 ALOX15 (0.50) KDM4EMAPTHPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750701-A Heterocyclic ethanolamine derivatives with β-adrenoreceptor agonistic activity SMITHKLINE BEECHAM PLC (GB) 1998-05-12 US disclosed
EP-0750617-A1 NOVEL HETEROCYCLIC ETHANOLAMINE DERIVATIVES WITH BETA-ADRENORECEPTOR AGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1997-01-02 EP disclosed
WO-1995025104-A1 NOVEL HETEROCYCLIC ETHANOLAMINE DERIVATIVES WITH BETA-ADRENORECEPTOR AGONISTIC ACTIVITY SMITHKLINE BEECHAM P.L.C. (GB) 1995-09-21 WO disclosed