SCHEMBL8620867

SCHEMBL8620867

CC(=O)Nc1c([N+](=O)[O-])cc([N+](=O)[O-])c2c1CCCC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.48
GAA P10253 3/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 4/20 0.45
HTT P42858 2/20 0.41
NPSR1 Q6W5P4 2/20 0.40
POLB P06746 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GALR2 O43603 1/20 0.38
MITF O75030 1/20 0.38
HSP90AA1 P07900 1/20 0.38
XBP1 P17861 1/20 0.38
CCR6 P51684 1/20 0.38
SLC9A1 P19634 1/20 0.38
DYRK1A Q13627 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26529166 0.88 MAPT (0.43) MAPTGAAKDM4ELMNAHTT
SCHEMBL6842000 0.79 MAPT (0.43) MAPTGAAKDM4ELMNAHTT
SCHEMBL8623539 0.79 ALDH1A1 (0.50) MAPTLMNAHTTNPSR1POLB
SCHEMBL2249641 0.77 HTT (0.49) MAPTGAALMNAHTTPOLB
SCHEMBL7154811 0.76 MAPT (0.50) MAPTGAALMNAHTTNPSR1
SCHEMBL2247139 0.75 HTT (0.48) MAPTGAALMNAHTTPOLB
SCHEMBL9362588 0.74 ALDH1A1 (0.38) MAPTGAAKDM4ELMNAHTT
SCHEMBL5203453 0.74 GAA (0.56) MAPTGAAKDM4ELMNAHTT
SCHEMBL28836799 0.74 GPR35 (0.55) MAPTGAAKDM4ELMNAHTT
SCHEMBL2246833 0.74 HTT (0.49) MAPTGAALMNAHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849744-A Pyrrolyl tetrahydrobenzoquinoxaline diones, their preparation and use as glutamate receptor antagonist BASF AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed