SCHEMBL8620870

SCHEMBL8620870

COc1cc2nccc(C(=O)NC(N)=Nc3ccccc3)c2cc1OC

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRC P12931 3/20 0.47
TGFBR1 P36897 3/20 0.47
PDGFRA P16234 5/20 0.46
KDR P35968 5/20 0.46
KIT P10721 4/20 0.46
SMO Q99835 1/20 0.45
PSMD14 O00487 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
RAB9A P51151 1/20 0.44
MET P08581 4/20 0.44
AURKA O14965 3/20 0.44
LCK P06239 3/20 0.44
TEK Q02763 3/20 0.44
AURKB Q96GD4 3/20 0.44
NUDT1 P36639 2/20 0.43
AXL P30530 1/20 0.43
ABL1 P00519 1/20 0.43
LYN P07948 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620947 0.86 KDM4E (0.60) NPC1LMNARAB9A
SCHEMBL8616502 0.86 KDM4E (0.48) PDGFRAKDRNPC1LMNARAB9A
SCHEMBL8613207 0.84 SMO (0.49) SMOPSMD14NPC1LMNARAB9A
SCHEMBL8619835 0.84 SMO (0.49) SMOPSMD14NPC1LMNARAB9A
SCHEMBL8617725 0.83 PDE4A (0.46) SMOPSMD14NPC1LMNARAB9A
SCHEMBL8620636 0.83 NPC1 (0.49) TGFBR1SMOPSMD14NPC1LMNA
SCHEMBL8612700 0.83 KDM4E (0.45) PDGFRAKDRLMNAMETAURKA
SCHEMBL8617741 0.82 SCN2A (0.44) NPC1LMNARAB9A
SCHEMBL8613854 0.82 SCN2A (0.44) NPC1LMNARAB9A
SCHEMBL8616307 0.82 SMO (0.43) SMOPSMD14NPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed