SCHEMBL8621073

SCHEMBL8621073

CCc1cc2c(cc1OC(=O)c1ccccc1)CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](OC(=O)COC(=O)CCCc3ccc(N(CCCl)CCCl)cc3)CC[C@@H]12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.46
KMT2A Q03164 7/20 0.46
LMNA P02545 7/20 0.46
CYP3A4 P08684 6/20 0.46
ESR1 P03372 6/20 0.46
MEN1 O00255 5/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
ADORA3 P0DMS8 4/20 0.46
TP53 P04637 4/20 0.46
ALOX15 P16050 3/20 0.46
ATM Q13315 2/20 0.46
PGR P06401 2/20 0.46
AR P10275 2/20 0.46
PTGS1 P23219 2/20 0.46
PDE3A Q14432 2/20 0.46
POLB P06746 1/20 0.46
CHRM1 P11229 1/20 0.46
TBXA2R P21731 1/20 0.46
USP2 O75604 1/20 0.46
NR3C1 P04150 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619814 0.92 LMNA (0.44) MAPTKMT2ALMNACYP3A4ESR1
Atrimustine SCHEMBL8659 0.90 LMNA (0.56) MAPTKMT2ALMNACYP3A4ESR1
Atrimustine SCHEMBL10580413 0.90 LMNA (0.56) MAPTKMT2ALMNACYP3A4ESR1
Atrimustine SCHEMBL29359877 0.90 LMNA (0.56) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL8619573 0.89 MAPT (0.41) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL8617441 0.87 MAPT (0.41) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL8619920 0.86 MAPT (0.39) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL8615788 0.85 KMT2A (0.44) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL10406599 0.85 LMNA (0.63) MAPTKMT2ALMNACYP3A4ESR1
SCHEMBL8621923 0.84 MAPT (0.38) MAPTKMT2ALMNACYP3A4ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573977-B1 Novel estradiol derivative-chlorambucil conjugate, process for preparing the same, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 1998-05-13 EP disclosed