SCHEMBL8621153

SCHEMBL8621153

CCc1cc(C#N)ccc1CNc1c(NC(C)C)c(=O)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.54
ABCC8 Q09428 1/20 0.54
KCNJ11 Q14654 1/20 0.54
KCNJ8 Q15842 1/20 0.54
KDM4C Q9H3R0 1/20 0.33
CYP2A6 P11509 1/20 0.33
SETDB1 Q15047 1/20 0.32
CXCR2 P25025 3/20 0.32
P2RX7 Q99572 1/20 0.32
EGLN2 Q96KS0 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32
LRRK2 Q5S007 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ELANE P08246 1/20 0.31
IDH1 O75874 4/20 0.31
ERBB2 P04626 1/20 0.31
PRKACA P17612 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887074 0.88 ABCC9 (0.71) ABCC9ABCC8KCNJ11KCNJ8RPS6KB1
SCHEMBL7895223 0.82 ABCC9 (0.51) ABCC9ABCC8KCNJ11KCNJ8KDM4C
SCHEMBL7887121 0.82 ABCC9 (0.43) ABCC9ABCC8KCNJ11KCNJ8KDM4C
SCHEMBL7898502 0.80 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8KDM4C
SCHEMBL7894087 0.79 LOXL2 (0.50) ABCC9ABCC8KCNJ11KCNJ8CYP2A6
SCHEMBL7895748 0.75 ABCC9 (0.61) ABCC9ABCC8KCNJ11KCNJ8IDH1
SCHEMBL7895591 0.74 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL7895113 0.74 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8P2RX7
SCHEMBL8414670 0.74 LRRK2 (0.42) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL13824727 0.73 CYP2A6 (0.52) ABCC9ABCC8KCNJ11KCNJ8KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US claimed
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US disclosed