SCHEMBL8624080

SCHEMBL8624080

COc1ccc(SSc2ccc(OC)cc2C=O)c(C=O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.59
ALDH1A1 P00352 8/20 0.56
TRIM24 O15164 1/20 0.55
TYR P14679 1/20 0.55
TRIM33 Q9UPN9 1/20 0.55
CYP1A2 P05177 4/20 0.47
KDM4E B2RXH2 3/20 0.47
CYP2C19 P33261 2/20 0.47
MAPT P10636 1/20 0.47
CYP2A6 P11509 1/20 0.45
LMNA P02545 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
JUN P05412 1/20 0.41
NFKB1 P19838 1/20 0.41
NFE2L2 Q16236 1/20 0.41
PRKDC P78527 1/20 0.40
RAB9A P51151 1/20 0.40
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7879327 0.86 ERN1 (0.50) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL30138984 0.81 ERN1 (0.56) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL16495093 0.80 ERN1 (0.50) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL12672585 0.79 ALDH1A1 (0.70) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL29957021 0.79 ALDH1A1 (0.70) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL6763816 0.79 ERN1 (0.49) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL16494291 0.77 ERN1 (0.47) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL11071247 0.76 ERN1 (0.46) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL4438653 0.76 ERN1 (0.50) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL2505574 0.76 ERN1 (0.63) ERN1ALDH1A1TRIM24TYRTRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10045706-A None JP disclosed
US-7393652-B2 Methods for identifying a chemical compound that directly enhances binding of FKBP12.6 to PKA-phosphorylated type 2 ryanodine receptor (RyR2) THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2008-07-01 US disclosed
JP-H1045706-A MEW DISULFIDE COMPOUND, PRODUCTION THEREOF AND PRODUCTION OF THIAZEPINE DERIVATIVE BY USING THE SAME COMPOUND SUMITOMO SEIKA CHEM CO LTD 1998-02-17 JP disclosed