SCHEMBL8624202

SCHEMBL8624202

COc1cccc(CC/C(C)=C/CCCC(P(=O)(O)O)S(=O)(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
FDFT1 P37268 1/20 0.37
CASP3 P42574 1/20 0.37
CASP7 P55210 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8624208 1.00 MTNR1A (0.41) MTNR1AMTNR1BHDAC1HDAC6AKR1C3
SCHEMBL8624172 0.86 FDPS (0.36) FNTAFNTB
SCHEMBL27415442 0.85 FNTA (0.34) FNTAFNTBFDFT1
SCHEMBL27395211 0.85 FDPS (0.36) FNTAFNTB
SCHEMBL8621102 0.85 ANPEP (0.40)
SCHEMBL8621107 0.85 ANPEP (0.40)
SCHEMBL8621189 0.85 ANPEP (0.40)
SCHEMBL27416174 0.84 ANPEP (0.39)
SCHEMBL27396721 0.84 ANPEP (0.39)
SCHEMBL8620707 0.83 FNTA (0.53) HDAC1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712396-A PHOSPHONOSULFONATE COMPOUNDS USED FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND ATHEROSCLEROSIS MAGNIN DAVID R (US) 1998-01-27 US disclosed
US-5567841-A ANTICHOLESTEROL AGENT BRISTOL-MYERS SQUIBB COMPANY (US) 1996-10-22 US disclosed
US-5470845-A Methods of using α-phosphonosulfonate squalene synthetase inhibitors including the treatment of atherosclerosis and hypercholesterolemia BRISTOL-MYERS SQUIBB COMPANY (US) 1995-11-28 US disclosed
EP-0595635-A1 Alpha-phosphorous substituted sulfonate derivatives as squalene synthetase inhibitors E.R. Squibb & Sons, Inc. (US) 1994-05-04 EP disclosed