SCHEMBL8624410

SCHEMBL8624410

CCOC(=O)/C=C(/C(=O)OCC)N(c1ccc(F)c(F)c1)C1CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
NPSR1 Q6W5P4 2/20 0.35
OPRD1 P41143 1/20 0.35
PTGIR P43119 2/20 0.34
PTGDR Q13258 1/20 0.34
NPY2R P49146 1/20 0.33
CHRM1 P11229 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 2/20 0.32
TSHR P16473 1/20 0.32
KCNN4 O15554 1/20 0.32
TACR1 P25103 2/20 0.32
SLC6A4 P31645 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628958 1.00 ALDH1A1 (0.38) ALDH1A1NPSR1OPRD1PTGIRPTGDR
SCHEMBL8627403 0.90 TACR1 (0.38) ALDH1A1PTGIRLMNACYP2C9KMT2A
SCHEMBL8624620 0.90 TACR1 (0.38) ALDH1A1PTGIRLMNACYP2C9KMT2A
SCHEMBL8622686 0.82 NPSR1 (0.35) ALDH1A1NPSR1MEN1LMNACYP1A2
SCHEMBL8626616 0.82 NPSR1 (0.35) ALDH1A1NPSR1MEN1LMNACYP1A2
SCHEMBL8624667 0.81 NPSR1 (0.39) ALDH1A1NPSR1MEN1LMNACYP1A2
SCHEMBL8621807 0.81 NPSR1 (0.39) ALDH1A1NPSR1MEN1LMNACYP1A2
SCHEMBL8624411 0.77 OPRD1 (0.39) ALDH1A1OPRD1PTGIRPTGDRNPY2R
SCHEMBL8645991 0.76 MEN1 (0.41) ALDH1A1NPSR1PTGIRPTGDRCHRM1
SCHEMBL31453592 0.72 ALDH1A1 (0.40) ALDH1A1PTGIRNPY2RLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
EP-0684942-A4 1995-12-27 EP disclosed
EP-0684942-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1995-12-06 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed
WO-1994019312-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1994-09-01 WO disclosed