SCHEMBL8625558

SCHEMBL8625558

CCOC(=O)C(=CN(c1ccc(F)c(F)c1F)C1CC1)C(=O)OCC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.40
MEN1 O00255 4/20 0.40
MAPT P10636 4/20 0.40
LMNA P02545 4/20 0.40
NPSR1 Q6W5P4 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
P2RX7 Q99572 2/20 0.35
S1PR4 O95977 1/20 0.35
S1PR1 P21453 1/20 0.35
MAPK1 P28482 1/20 0.35
EPHX2 P34913 2/20 0.34
DHODH Q02127 2/20 0.34
GAA P10253 3/20 0.33
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
PLIN1 O60240 1/20 0.33
POLB P06746 1/20 0.33
PLIN5 Q00G26 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651194 0.92 MAPT (0.39) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL6647935 0.89 NPSR1 (0.37) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL6653250 0.86 MEN1 (0.35) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL8645991 0.81 MEN1 (0.41) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL25069399 0.81 NPSR1 (0.40) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL8622781 0.80 KMT2A (0.43) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL8626320 0.79 ALDH1A1 (0.40) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL10656978 0.78 KMT2A (0.42) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL262000 0.77 MAPT (0.38) KMT2AMEN1MAPTLMNANPSR1
SCHEMBL8625478 0.77 KMT2A (0.41) KMT2AMEN1MAPTLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
EP-0684942-A4 1995-12-27 EP disclosed
EP-0684942-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1995-12-06 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed
WO-1994019312-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1994-09-01 WO disclosed