SCHEMBL8626508

SCHEMBL8626508

CCCCn1c(S)nnc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RGS4 P49798 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11691595 0.76 SMN1; SMN2 (0.42) TSHRLMNAALDH1A1
SCHEMBL16774865 0.72 TLR8 (0.39) TSHRLMNAHTTKDM4EALDH1A1
SCHEMBL5657269 0.69 TSHR (0.36) TSHRRGS4
SCHEMBL11381038 0.69 ALDH1A1 (0.38) TSHRALDH1A1RGS4
SCHEMBL8173050 0.68 TSHR (0.35) TSHRLMNAALDH1A1
SCHEMBL14342088 0.67 HSD11B1 (0.41) TSHRLMNAHTTALDH1A1
SCHEMBL15166513 0.67 HSD11B1 (0.41)
SCHEMBL11512011 0.67 HSD11B1 (0.41) TSHRLMNAHTTALDH1A1
SCHEMBL14557069 0.67 HSD11B1 (0.41) TSHRLMNAHTTALDH1A1
SCHEMBL9642497 0.67 TLR8 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed