SCHEMBL8627596

SCHEMBL8627596

CCCCC1=NS(=O)(=O)c2cnccc2N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.41
LMNA P02545 4/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
THRB P10828 1/20 0.38
MAPT P10636 5/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36
MAPK1 P28482 2/20 0.36
POLB P06746 2/20 0.36
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8629245 0.90 ALDH1A1 (0.37) ALDH1A1LMNASMN1; SMN2THRBMAPT
SCHEMBL8627414 0.85 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2THRBMAPT
SCHEMBL8761102 0.78 ALDH1A1 (0.41) ALDH1A1LMNASMN1; SMN2THRBMAPT
SCHEMBL8626608 0.77 KDM6B (0.41) ALDH1A1LMNASMN1; SMN2CYP3A4CA12
SCHEMBL8761359 0.76 ALDH1A1 (0.45) ALDH1A1LMNASMN1; SMN2MAPTNPC1
SCHEMBL6619663 0.76 LATS1 (0.40) LMNASMN1; SMN2POLBKDM4C
SCHEMBL719010 0.75 NPC1 (0.47) ALDH1A1LMNASMN1; SMN2THRBMAPT
SCHEMBL394795 0.75 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2THRBMAPT
SCHEMBL6618966 0.75 L3MBTL1 (0.32) ALDH1A1LMNASMN1; SMN2MAPTCYP1A2
SCHEMBL8286622 0.74 CA12 (0.62) ALDH1A1LMNASMN1; SMN2THRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed