SCHEMBL8628051

SCHEMBL8628051

COc1ccc(-c2c(-c3ccccc3S(N)(=O)=O)nn(CCN(C)C)c2C(F)(F)F)cc1C

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.41
PTGS1 P23219 4/20 0.41
F10 P00742 6/20 0.38
P2RX3 P56373 3/20 0.37
BRD4 O60885 1/20 0.35
SLC6A9 P48067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635102 0.92 PTGS2 (0.43) PTGS2PTGS1F10P2RX3
SCHEMBL8629957 0.89 PTGS2 (0.48) PTGS2PTGS1F10P2RX3
SCHEMBL8634283 0.88 F10 (0.42) PTGS2PTGS1F10P2RX3
SCHEMBL8633042 0.87 PTGS2 (0.41) PTGS2PTGS1F10
SCHEMBL8631636 0.87 F10 (0.46) PTGS2PTGS1F10
SCHEMBL8630046 0.86 PTGS2 (0.42) PTGS2PTGS1F10
SCHEMBL7780086 0.86 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8629728 0.86 PTGS2 (0.44) PTGS2PTGS1F10
SCHEMBL8634387 0.86 PTGS2 (0.46) PTGS2PTGS1F10P2RX3BRD4
SCHEMBL8635364 0.85 PTGS2 (0.44) PTGS2PTGS1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed