SCHEMBL8628608

SCHEMBL8628608

N#Cc1ccc(S(=O)(=O)Nc2cccnc2Nc2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 3/20 0.61
TUBB4A P04350 1/20 0.55
TUBB P07437 1/20 0.55
TUBA3C P0DPH7 1/20 0.55
TUBA1B P68363 1/20 0.55
TUBA4A P68366 1/20 0.55
TUBB4B P68371 1/20 0.55
TUBB3 Q13509 1/20 0.55
TUBB2A Q13885 1/20 0.55
TUBB8 Q3ZCM7 1/20 0.55
TUBA3E Q6PEY2 1/20 0.55
TUBA1A Q71U36 1/20 0.55
TUBA1C Q9BQE3 1/20 0.55
TUBB6 Q9BUF5 1/20 0.55
TUBB2B Q9BVA1 1/20 0.55
TUBB1 Q9H4B7 1/20 0.55
HSD11B1 P28845 3/20 0.54
SLC22A12 Q96S37 3/20 0.50
CYP19A1 P11511 1/20 0.49
AR P10275 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006004 0.87 TUBB4A (0.60) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8623534 0.85 KMT2A (0.60) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8623823 0.84 TUBB4A (0.61) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8623512 0.84 TUBB4A (0.74) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8623477 0.84 SLC40A1 (0.59) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8626115 0.81 TUBB4A (0.65) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8622659 0.81 TUBB4A (0.64) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8625569 0.81 MAPK1 (0.63) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8625500 0.81 TUBB4A (0.57) GLO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8623536 0.81 TUBB4A (0.81) GLO1TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP disclosed
US-5610304-A Pyrimidinyl or pyridinyl sulfonamide substituted compounds EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5434172-A Antitumor EISAI CO., LTD. (JP) 1995-07-18 US disclosed
US-5332751-A Antitumor EISAI CO., LTD. (JP) 1994-07-26 US disclosed
US-5292758-A Sulfonamide derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5250549-A Antitumor agents EISAI CO., LTD. (JP) 1993-10-05 US disclosed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP disclosed