SCHEMBL8628901

SCHEMBL8628901

OCC1Cc2ccccc2C=N1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.35
HTR2B P41595 1/20 0.32
IDO1 P14902 2/20 0.31
CYP19A1 P11511 2/20 0.30
KDM4E B2RXH2 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28139657 1.00 TRPA1 (0.35) TRPA1HTR2BIDO1CYP19A1KDM4E
SCHEMBL31168159 1.00 TRPA1 (0.35) TRPA1HTR2BIDO1CYP19A1KDM4E
SCHEMBL28188526 0.86 TRPA1 (0.37) TRPA1
SCHEMBL28139052 0.81 PNMT (0.37) TRPA1IDO1CYP19A1KDM4EL3MBTL1
SCHEMBL7508347 0.81 KDM4E (0.36) TRPA1IDO1CYP19A1KDM4EL3MBTL1
SCHEMBL28139649 0.81 HTR2A (0.36) TRPA1IDO1CYP19A1KDM4EL3MBTL1
SCHEMBL28853799 0.79 HTR2A (0.40) TRPA1IDO1
SCHEMBL28188528 0.77 TRPA1 (0.33) TRPA1
SCHEMBL29914779 0.76 PNMT (0.42)
SCHEMBL27159819 0.76 PNMT (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064493-A1 COMPOUNDS AND METHODS FOR TREATING CORONAVIRUSES Clear Creek Bio, Inc. (US) 2023-04-20 WO disclosed
CN-110049780-A Isoquinolinebenzodiazepine (IQB) -1 (chloromethyl) -2, 3-dihydro-1H-benzo [ E ] indole (CBI) dimer 塞勒兰特治疗公司 2019-07-23 CN disclosed
US-5780589-A DIPEPTIDES, TRIPEPTIDES OR CYCLIC PEPTIDES AS ANTAGONIST OF OPIOID RECEPTORS TREATING DRUG ABUSE, DRUG DEPENDENCE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-07-14 US disclosed