SCHEMBL8628903

SCHEMBL8628903

COC(=O)C#CC(=O)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
GSK3B P49841 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
ERCC5 P28715 1/20 0.42
FEN1 P39748 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
MAOB P27338 2/20 0.41
PTGS2 P35354 2/20 0.41
MAOA P21397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10428831 0.83 CA1 (0.53) HPGDALDH1A1HTTLMNAMAPT
SCHEMBL8627919 0.83 TDP1 (0.53) HPGDCES2CES1GSK3BALDH1A1
SCHEMBL8626139 0.81 APP (0.55) CES2CES1GSK3BALDH1A1ALOX15
SCHEMBL10428885 0.81 APP (0.47) CES2CES1HTTALOX15TSHR
SCHEMBL3198121 0.81 TSHR (0.52) HPGDCES2CES1ALDH1A1ALOX15
SCHEMBL8625862 0.81 HPGD (0.49) HPGDHTTTSHRKDM4EMAPT
SCHEMBL8630144 0.80 ERCC5 (0.47) HPGDALDH1A1ERCC5FEN1
SCHEMBL10429071 0.79 APP (0.53) HPGDALDH1A1HTTTSHRKDM4E
SCHEMBL10428960 0.79 PLK1 (0.49) HPGDALDH1A1HTTALOX15TSHR
SCHEMBL27978391 0.79 SMN1; SMN2 (0.42) HPGDALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646570-B1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO (JP) 1998-06-24 EP disclosed
US-5488134-A Preparation of compounds of lignan series SHIONOGI & CO., LTD. (JP) 1996-01-30 US disclosed
EP-0646570-A1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO., LTD. (JP) 1995-04-05 EP disclosed
US-4929741-A ANTISECRETORY AGENTS, GASTRIC JUICE, ANTIULCER AGENTS HOFFMAN-LA ROCHE INC. (US) 1990-05-29 US disclosed
EP-0282898-A2 Propiolophenone derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-09-21 EP disclosed