SCHEMBL8628980

SCHEMBL8628980

Cc1cc(N)ccc1C(=O)N1CC(OCCCN2CCCC2)CCc2cc(F)ccc21

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.47
PDK1 Q15118 4/20 0.38
PDK2 Q15119 4/20 0.38
PDK3 Q15120 4/20 0.38
PDK4 Q16654 4/20 0.38
CHRM1 P11229 1/20 0.37
DRD2 P14416 3/20 0.37
HTR2A P28223 2/20 0.37
HTR7 P34969 1/20 0.37
HRH1 P35367 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
NOTUM Q6P988 1/20 0.35
HSP90AA1 P07900 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL8634376 0.87 KDM4E (0.38) PDK1PDK2PDK3PDK4HTR7
SCHEMBL8628984 0.85 AVPR2 (0.46) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL4685307 0.81 AVPR2 (0.45) AVPR2HTR7HRH1HRH3
SCHEMBL8628978 0.81 AVPR2 (0.47) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL4682848 0.75 AVPR2 (0.45) AVPR2HTR7HRH3
SCHEMBL8629473 0.74 AVPR2 (0.51) AVPR2NOTUM
SCHEMBL8628399 0.74 ALDH1A1 (0.37) HTR7
SCHEMBL8630394 0.72 ALDH1A1 (0.34) PDK1PDK2PDK3PDK4HSP90AA1
Iodide SCHEMBL8634378 0.72 ALDH1A1 (0.37) PDK1PDK2PDK3PDK4HTR7
SCHEMBL8632568 0.72 AVPR2 (0.43) AVPR2CHRM1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed