SCHEMBL8628978

SCHEMBL8628978

CCC(OC1CCc2cc(F)ccc2N(C(=O)c2ccc(N)cc2C)C1)N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.47
PDK1 Q15118 6/20 0.38
PDK2 Q15119 6/20 0.38
PDK3 Q15120 6/20 0.38
PDK4 Q16654 6/20 0.38
NOTUM Q6P988 1/20 0.35
HSP90AA1 P07900 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.33
HTT P42858 2/20 0.33
KCNQ2 O43526 1/20 0.33
HSD11B1 P28845 1/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL8634375 0.87 MAPT (0.37) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL8628980 0.81 AVPR2 (0.47) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL8628397 0.74 IDO1 (0.33) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL8629470 0.71 AVPR2 (0.50) AVPR2LMNA
SCHEMBL8628984 0.68 AVPR2 (0.46) AVPR2PDK1PDK2PDK3PDK4
Iodide SCHEMBL8634376 0.68 KDM4E (0.38) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL8628503 0.65 AVPR2 (0.39) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL8634049 0.65 AVPR2 (0.42) AVPR2
SCHEMBL8629473 0.65 AVPR2 (0.51) AVPR2NOTUMLMNA
SCHEMBL4685307 0.65 AVPR2 (0.45) AVPR2TSHRALDH1A1HTTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed