SCHEMBL8629049

SCHEMBL8629049

N#Cc1cccc(CN2CCC(OS(=O)(=O)c3cccs3)C2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
ALDH1A1 P00352 4/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FEN1 P39748 1/20 0.37
POLB P06746 2/20 0.36
MAPK8 P45983 1/20 0.36
DPP4 P27487 1/20 0.36
FAP Q12884 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
CHRM3 P20309 1/20 0.36
KCNH2 Q12809 2/20 0.36
MMP1 P03956 1/20 0.36
ADAM17 P78536 1/20 0.36
F10 P00742 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628686 0.87 KCNH2 (0.40) ROCK2ROCK1SIRT2SIRT1ALDH1A1
SCHEMBL8625901 0.83 F10 (0.52) ROCK2ROCK1SIRT2SIRT1ALDH1A1
SCHEMBL8622748 0.79 F10 (0.43) ROCK2ROCK1KCNH2F10FNTA
SCHEMBL8622746 0.79 KCNH2 (0.40) ROCK2ROCK1ALDH1A1PKMSMN1; SMN2
SCHEMBL8624162 0.79 F10 (0.54) ROCK2ROCK1ALDH1A1KCNH2F10
SCHEMBL7423237 0.73 FNTA (0.51) ROCK2ROCK1SIRT2SIRT1ALDH1A1
SCHEMBL7482530 0.72 SIRT2 (0.48) ROCK2ROCK1SIRT2SIRT1DPP4
SCHEMBL12009728 0.72 SIRT2 (0.46) ROCK2ROCK1SIRT2SIRT1ALDH1A1
SCHEMBL7419120 0.72 SIRT2 (0.48) ROCK2ROCK1SIRT2SIRT1DPP4
SCHEMBL8423834 0.71 F10 (0.41) SIRT2SIRT1ALDH1A1DPP4FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731315-A Substituted sulfonic acid n- (aminoiminomethyl)phenylalkyl!-azaheterocyclamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-03-24 US disclosed