SCHEMBL8629917

SCHEMBL8629917

CCOC(=O)Cn1nc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.72
PTGS1 P23219 2/20 0.61
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
GAA P10253 1/20 0.49
CA9 Q16790 4/20 0.48
CA12 O43570 3/20 0.48
TRPM2 O94759 1/20 0.47
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MT-CO2 P00403 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
LMNA P02545 1/20 0.43
CA3 P07451 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634891 0.93 PTGS2 (0.73) PTGS2PTGS1CA9CA12TRPM2
SCHEMBL8633238 0.92 PTGS2 (0.84) PTGS2PTGS1GAACA9CA12
SCHEMBL8631631 0.91 PTGS2 (0.70) PTGS2PTGS1CA9CA12TRPM2
SCHEMBL8632520 0.91 PTGS2 (0.85) PTGS2PTGS1MEN1KMT2AGAA
SCHEMBL8630457 0.91 PTGS2 (0.69) PTGS2PTGS1CA9CA12TRPM2
SCHEMBL8635122 0.90 PTGS2 (0.68) PTGS2PTGS1MEN1KMT2ACA9
SCHEMBL8632389 0.90 PTGS2 (0.63) PTGS2PTGS1MEN1KMT2AGAA
SCHEMBL8631062 0.87 PTGS2 (0.67) PTGS2PTGS1CA9CA12TRPM2
SCHEMBL7780571 0.87 PTGS2 (0.63) PTGS2PTGS1CA9CA1CA2
SCHEMBL8631373 0.86 PTGS2 (0.63) PTGS2PTGS1CA9CA12TRPM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed