SCHEMBL8630628

SCHEMBL8630628

COC1CC(OCC(=O)NCCN2CCOCC2)c2cc(Cl)ccc2N(C(=O)c2ccc(NC(=O)c3ccccc3Br)cc2)C1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 15/20 0.47
EPHX2 P34913 2/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
AVPR1A P37288 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4684464 0.81 AVPR2 (0.49) AVPR2HTTMEN1ALDH1A1CYP1A2
SCHEMBL8630292 0.77 AVPR2 (0.43) AVPR2ALDH1A1CYP2C9AVPR1A
SCHEMBL8630692 0.76 AVPR2 (0.43) AVPR2ALDH1A1CYP2C9AVPR1A
SCHEMBL4685002 0.75 AVPR2 (0.46) AVPR2MEN1ALDH1A1KMT2AAVPR1A
SCHEMBL8715447 0.71 AVPR1A (0.53) AVPR2CYP2C9AVPR1A
SCHEMBL8712407 0.70 AVPR2 (0.52) AVPR2AVPR1A
SCHEMBL8628740 0.70 AVPR2 (0.48) AVPR2AVPR1A
SCHEMBL8713758 0.69 AVPR1A (0.53) AVPR2CYP2C9AVPR1A
Hydrochloric Acid SCHEMBL8630729 0.69 AVPR2 (0.48) AVPR2CYP2C9AVPR1A
SCHEMBL8632029 0.69 AVPR2 (0.48) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed