SCHEMBL8630692

SCHEMBL8630692

COC1CC(CC(=O)N2CCN(C)CC2)c2cc(Cl)ccc2N(C(=O)c2ccc(NC(=O)c3ccccc3Br)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 12/20 0.43
AVPR1A P37288 9/20 0.43
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2C9 P11712 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
ABCB11 O95342 1/20 0.39
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
TBXA2R P21731 1/20 0.39
HTR2C P28335 1/20 0.39
HRH1 P35367 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632029 0.92 AVPR2 (0.48) AVPR2AVPR1AABCB11ADRB2HTR1A
Hydrochloric Acid SCHEMBL8630729 0.92 AVPR2 (0.48) AVPR2AVPR1ACYP2C9ABCB11ADRB2
SCHEMBL8630292 0.87 AVPR2 (0.43) AVPR2AVPR1ACYP2C9USP2ALDH1A1
SCHEMBL8628740 0.79 AVPR2 (0.48) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL4683086 0.79 AVPR2 (0.46) AVPR2AVPR1ASMN1; SMN2USP2ALDH1A1
Hydrochloric Acid SCHEMBL4681785 0.78 AVPR2 (0.51) AVPR2AVPR1AABCB11ADRB2HTR1A
Hydrochloric Acid SCHEMBL4687939 0.78 AVPR2 (0.60) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL8630759 0.78 AVPR1A (0.47) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL4687153 0.77 AVPR2 (0.48) AVPR2AVPR1ASMN1; SMN2USP2ALDH1A1
SCHEMBL8631280 0.77 AVPR2 (0.49) AVPR2AVPR1AABCB11ADRB2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed