SCHEMBL8630759

SCHEMBL8630759

COC1CC(CC(=O)N2CCCCC2)c2cc(F)ccc2N(C(=O)c2ccc(NC(=O)c3ccccc3C)cc2)C1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 7/20 0.47
AVPR2 P30518 6/20 0.47
OXTR P30559 2/20 0.45
AVPR1B P47901 2/20 0.45
ABCB11 O95342 1/20 0.45
HTR1A P08908 1/20 0.45
CHRM1 P11229 1/20 0.45
SLC6A4 P31645 1/20 0.45
ADRA1A P35348 1/20 0.45
OPRM1 P35372 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681827 0.86 AVPR2 (0.60) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL8632029 0.85 AVPR2 (0.48) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL8629514 0.83 AVPR2 (0.44) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL7353320 0.79 AVPR2 (0.55) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL8628740 0.79 AVPR2 (0.48) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL8630756 0.79 AVPR1A (0.46) AVPR1AAVPR2OXTRAVPR1BABCB11
SCHEMBL7336268 0.79 AVPR2 (0.50) AVPR1AAVPR2OXTRAVPR1BABCB11
Hydrochloric Acid SCHEMBL8630729 0.78 AVPR2 (0.48) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL8630692 0.78 AVPR2 (0.43) AVPR1AAVPR2ABCB11HTR1ACHRM1
SCHEMBL8631280 0.77 AVPR2 (0.49) AVPR1AAVPR2OXTRAVPR1BABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed