SCHEMBL8630930

SCHEMBL8630930

CC(=O)c1c(S(=O)(=O)N(C)c2ccccc2)ccc(C)c1N1CCN(c2ccncc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.39
LMNA P02545 3/20 0.39
CTDSP1 Q9GZU7 1/20 0.38
MAPK1 P28482 2/20 0.37
TSHR P16473 1/20 0.37
PKM P14618 2/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 2/20 0.36
KDM4E B2RXH2 2/20 0.36
HTR1A P08908 4/20 0.36
HTR2A P28223 2/20 0.36
CLEC4M Q9H2X3 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RECQL P46063 1/20 0.35
CA12 O43570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696712 0.87 ESR1 (0.45) SMN1; SMN2CTDSP1MAPK1TSHRMEN1
SCHEMBL8637224 0.83 POLB (0.38) SMN1; SMN2LMNACTDSP1TSHRPKM
SCHEMBL8634739 0.69 CA12 (0.41) LMNAMEN1KMT2AMAPTGAA
SCHEMBL8697322 0.66 MAPT (0.36) SMN1; SMN2LMNAMAPTGAAKDM4E
SCHEMBL8634709 0.64 CYP1A2 (0.36) SMN1; SMN2MAPK1TSHRMAPTGAA
SCHEMBL20036118 0.64 PKM (0.51) SMN1; SMN2LMNAMAPK1TSHRPKM
SCHEMBL27350346 0.64 MAPT (0.55) LMNAMAPK1MEN1KMT2AMAPT
SCHEMBL11673375 0.62 CHKA (0.63) SMN1; SMN2LMNATSHRMEN1ALOX15
SCHEMBL18590696 0.62 CHKA (0.67) SMN1; SMN2LMNAMAPTGAAKDM4E
SCHEMBL7956272 0.61 NPC1 (0.69) SMN1; SMN2TSHRMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed