SCHEMBL8630959

SCHEMBL8630959

CC(=O)OC(c1ccccc1)c1scnc1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GLS O94925 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
PABPC1 P11940 1/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
TSHR P16473 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
CYP19A1 P11511 2/20 0.34
P2RX7 Q99572 2/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026489 0.96 SLC6A3 (0.39) ALDH1A1CYP3A4SLC6A3KDM4EPKM
SCHEMBL9025789 0.94 SLC6A3 (0.37) ALDH1A1CYP3A4SLC6A3KDM4EPKM
SCHEMBL14962416 0.85 SLC6A3 (0.41) ALDH1A1SLC6A3KDM4EPKMSMN1; SMN2
SCHEMBL14962415 0.82 SLC6A3 (0.39) CYP3A4SLC6A3KDM4EPKMHSD17B10
SCHEMBL14962413 0.82 SLC6A3 (0.39) CYP3A4SLC6A3KDM4EPKMHSD17B10
SCHEMBL8634186 0.81 MEN1 (0.41) P2RX7
SCHEMBL14962414 0.81 SLC6A3 (0.38) ALDH1A1SLC6A3KDM4EPKMSMN1; SMN2
SCHEMBL9025932 0.80 SLC6A3 (0.42) SLC6A3KDM4EPKMSMN1; SMN2TSHR
SCHEMBL12180158 0.78 SLC6A3 (0.39) SLC6A3KDM4EPKMSMN1; SMN2TSHR
SCHEMBL14962409 0.76 SLC6A3 (0.40) ALDH1A1SLC6A3KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed