SCHEMBL8631053

SCHEMBL8631053

COc1ccc(-c2c(-c3ccccc3S(N)(=O)=O)nn(CCc3ccccc3)c2C(F)(F)C(F)(F)F)cc1F

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.44
PTGS1 P23219 8/20 0.42
F10 P00742 4/20 0.39
P2RX3 P56373 4/20 0.36
PI4KB Q9UBF8 1/20 0.36
F2 P00734 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630480 0.92 PTGS2 (0.43) PTGS2PTGS1F10PI4KBF2
SCHEMBL8629097 0.89 PTGS2 (0.45) PTGS2PTGS1F10F2
SCHEMBL7777495 0.89 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8635624 0.88 PTGS2 (0.45) PTGS2PTGS1F10P2RX3PI4KB
SCHEMBL8632811 0.85 PTGS2 (0.43) PTGS2PTGS1F10P2RX3PI4KB
SCHEMBL8632921 0.85 PTGS2 (0.46) PTGS2PTGS1F10P2RX3PI4KB
SCHEMBL8630564 0.85 PTGS2 (0.45) PTGS2PTGS1F10PI4KBF2
SCHEMBL8632828 0.85 PTGS2 (0.49) PTGS2PTGS1F10P2RX3F2
SCHEMBL8634717 0.85 PTGS2 (0.43) PTGS2PTGS1F10P2RX3PI4KB
SCHEMBL7780078 0.84 PTGS2 (0.64) PTGS2PTGS1PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed