SCHEMBL8631456

SCHEMBL8631456

O=C(O)c1ccccc1N1CCN(c2ccncc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
TSHR P16473 2/20 0.49
MEN1 O00255 1/20 0.49
USP2 O75604 1/20 0.49
KMT2A Q03164 1/20 0.49
MLYCD O95822 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
CYP2C9 P11712 2/20 0.46
CHKA P35790 1/20 0.46
CYP2C19 P33261 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
ENPP2 Q13822 2/20 0.45
MYC P01106 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPK1 P28482 1/20 0.45
HIF1A Q16665 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3808106 0.89 ALDH1A1 (0.70) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL8630996 0.86 CHKA (0.44) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL10684394 0.86 NPC1 (0.62) ALDH1A1TSHRMEN1USP2KMT2A
Hydrochloric Acid SCHEMBL8632109 0.85 AKR1C3 (0.43) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL8048603 0.85 ALDH1A1 (0.61) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL8696589 0.84 CA12 (0.49) ALDH1A1TSHRMEN1KMT2ASMN1; SMN2
SCHEMBL15286530 0.83 CA12 (0.55) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL8544999 0.79 ALDH1A1 (0.55) ALDH1A1TSHRMEN1USP2KMT2A
SCHEMBL7236851 0.79 KMT2A (0.62) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL2492855 0.78 NPC1 (0.68) ALDH1A1TSHRUSP2SMN1; SMN2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed