SCHEMBL8696589

SCHEMBL8696589

O=C(O)c1cnccc1N1CCN(c2ccncc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.49
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA9 Q16790 3/20 0.49
CHKA P35790 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
CYP3A4 P08684 1/20 0.42
AKR1C3 P42330 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
ADRB2 P07550 1/20 0.42
NCF1 P14598 1/20 0.42
PLD1 Q13393 1/20 0.42
ALDH1A1 P00352 2/20 0.42
TRPV1 Q8NER1 1/20 0.42
ITGB3 P05106 3/20 0.41
ITGA2B P08514 3/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KDM6B O15054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631456 0.84 ALDH1A1 (0.56) CA12CA1CA2CA9CHKA
SCHEMBL4907976 0.84 SMN1; SMN2 (0.50) SMN1; SMN2CYP3A4CYP2C9TSHRALDH1A1
Potassium SCHEMBL30402396 0.83 SMN1; SMN2 (0.49) SMN1; SMN2CYP3A4CYP2C9TSHRALDH1A1
SCHEMBL398926 0.81 KDM4C (0.41) CA12CA1CA2CA9SMN1; SMN2
SCHEMBL15286530 0.80 CA12 (0.55) CA12CA1CA2CA9SMN1; SMN2
SCHEMBL8669300 0.76 GPR119 (0.53) ALDH1A1MEN1MAPTKMT2A
Biphenyl SCHEMBL27395942 0.76 HTR6 (0.48) CYP3A4ADRB2NCF1ALDH1A1
SCHEMBL30331023 0.76 F10 (0.39) CA12CA1CA2CA9CYP3A4
SCHEMBL7947516 0.75 KDM4E (0.59) CHKASMN1; SMN2CYP3A4AKR1C3CYP2C9
SCHEMBL10684394 0.74 NPC1 (0.62) CA12CA1CA2CA9CHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed