SCHEMBL8631780

SCHEMBL8631780

COc1cc(C(=O)N2c3ccc(Cl)cc3CCC(CCN3CCCCC3)C2OCC(N)=O)ccc1NC(=O)c1ccccc1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 1/20 0.38
AVPR1A P37288 2/20 0.38
AVPR2 P30518 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
AVPR1B P47901 1/20 0.37
PYGL P06737 1/20 0.36
GAA P10253 1/20 0.36
LMNA P02545 2/20 0.36
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
SPTLC2 O15270 1/20 0.35
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ABCB1 P08183 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631785 0.73 ABCB1 (0.38) ALDH1A1AVPR1AAVPR2LMNAESR1
SCHEMBL4685002 0.73 AVPR2 (0.46) ALDH1A1MAPTKDM4EAVPR1AAVPR2
SCHEMBL8632028 0.72 GRM4 (0.41) ALDH1A1KDM4EAVPR1AAVPR2KMT2A
SCHEMBL4687862 0.68 AVPR2 (0.47) ALDH1A1AVPR1AAVPR2MEN1KMT2A
SCHEMBL4684464 0.68 AVPR2 (0.49) ALDH1A1MAPTKDM4EAVPR1AAVPR2
SCHEMBL4683086 0.68 AVPR2 (0.46) ALDH1A1AVPR1AAVPR2MEN1KMT2A
SCHEMBL4687810 0.66 AVPR2 (0.48) ALDH1A1AVPR1AAVPR2AVPR1BPYGL
SCHEMBL4687283 0.66 AVPR2 (0.51) MAPTAVPR1AAVPR2MEN1KMT2A
SCHEMBL4687153 0.66 AVPR2 (0.48) ALDH1A1AVPR1AAVPR2MEN1KMT2A
SCHEMBL4687327 0.65 AVPR2 (0.55) MAPTAVPR1AAVPR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed