SCHEMBL8631785

SCHEMBL8631785

COC1CCc2cc(Cl)ccc2N(C(=O)c2ccc(NC(=O)c3ccccc3Br)cc2)C1(CCN1CCCCC1)OCC(N)=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
AVPR2 P30518 10/20 0.38
LMNA P02545 1/20 0.37
HSD11B1 P28845 2/20 0.37
AVPR1A P37288 5/20 0.36
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630006 0.77 AVPR2 (0.42) AVPR2LMNAHSD11B1AVPR1AALDH1A1
Hydrochloric Acid SCHEMBL8661682 0.73 LMNA (0.44) AVPR2LMNAHSD11B1AVPR1AALDH1A1
SCHEMBL8631780 0.73 ALDH1A1 (0.38) ABCB1ABCG2AVPR2LMNAAVPR1A
Hydrochloric Acid SCHEMBL8634039 0.73 LMNA (0.45) AVPR2LMNAHSD11B1AVPR1AALDH1A1
SCHEMBL8632078 0.70 AVPR1A (0.42) AVPR2LMNAHSD11B1AVPR1ATP53
SCHEMBL8632578 0.69 AVPR2 (0.44) AVPR2LMNAHSD11B1AVPR1ATP53
Hydrochloric Acid SCHEMBL8632564 0.69 AVPR2 (0.46) AVPR2AVPR1A
Hydrochloric Acid SCHEMBL8631933 0.68 AVPR2 (0.47) AVPR2LMNAAVPR1ATP53
SCHEMBL8634000 0.67 AVPR1A (0.41) AVPR2HSD11B1AVPR1A
Hydrochloric Acid SCHEMBL8632123 0.67 AVPR2 (0.45) AVPR2LMNAAVPR1ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed