SCHEMBL8631992

SCHEMBL8631992

CC(=O)C(OC1CCNCC1OCC(=O)O)(C(=O)O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.44
ITGA2B P08514 15/20 0.44
CYP2C9 P11712 2/20 0.34
TSHR P16473 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HRH3 Q9Y5N1 2/20 0.32
ADRB2 P07550 1/20 0.32
NCF1 P14598 1/20 0.32
PLD1 Q13393 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637046 0.81 ADRB2 (0.42) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8635510 0.79 RPLP1 (0.39) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8631565 0.69 ADRB2 (0.44) ITGB3ITGA2BCYP2C9TSHRCYP3A4
SCHEMBL8701123 0.69 ADRB2 (0.42) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8633634 0.69 CYP2C9 (0.46) ITGB3ITGA2BCYP2C9TSHRCYP3A4
Hydrochloric Acid SCHEMBL8838142 0.68 ADRB2 (0.41) ITGB3ITGA2BCYP2C9TSHRHRH3
Hydrochloric Acid SCHEMBL8838080 0.66 ADRB2 (0.53) ITGB3ITGA2BCYP2C9TSHRCYP3A4
SCHEMBL8632681 0.66 ADRB2 (0.43) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8636233 0.66 CHRM1 (0.39) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8634909 0.66 KDM4E (0.39) ITGB3ITGA2BCYP2C9TSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed