SCHEMBL8634909

SCHEMBL8634909

CC(=O)C(Oc1ccccc1C)(C(=O)O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
CHRM1 P11229 1/20 0.39
SLC2A1 P11166 4/20 0.38
CYP2C9 P11712 2/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 2/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
NPC1 O15118 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
HRH3 Q9Y5N1 3/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632213 0.89 SLC2A1 (0.43) KDM4EGAAMAPTCHRM1SLC2A1
SCHEMBL8635651 0.87 ALDH1A1 (0.46) KDM4EGAAMAPTCHRM1CYP2C9
SCHEMBL8633634 0.86 CYP2C9 (0.46) KDM4EGAAMAPTCYP2C9TSHR
SCHEMBL8631971 0.81 ITGB3 (0.40) KDM4EGAAMAPTSLC2A1CYP2C9
SCHEMBL8636233 0.80 CHRM1 (0.39) KDM4EGAAMAPTCHRM1SLC2A1
SCHEMBL8634772 0.79 GAA (0.39) KDM4EGAAMAPTCYP2C9TSHR
SCHEMBL8635770 0.78 ROCK2 (0.49) GAAMAPTCYP2C9TSHRALDH1A1
SCHEMBL8635264 0.77 CYP2C9 (0.44) KDM4EGAAMAPTCYP2C9TSHR
SCHEMBL8632705 0.76 CYP2C9 (0.42) KDM4EGAAMAPTCYP2C9TSHR
SCHEMBL8633523 0.75 AOC3 (0.38) MAPTCHRM1ALDH1A1MAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed