SCHEMBL8632237

SCHEMBL8632237

COC1CCC(OCCNCc2ccccc2)c2cc(Cl)ccc2N1C(=O)c1ccc(NC(=O)c2ccccc2Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 4/20 0.42
AVPR1A P37288 4/20 0.42
POLB P06746 1/20 0.39
PPARG P37231 2/20 0.39
HSD11B1 P28845 3/20 0.39
SMO Q99835 1/20 0.38
CHRM1 P11229 2/20 0.37
ABCB11 O95342 1/20 0.37
ADRB2 P07550 1/20 0.37
HTR1A P08908 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
TBXA2R P21731 1/20 0.37
HTR2C P28335 1/20 0.37
HRH1 P35367 1/20 0.37
OPRM1 P35372 1/20 0.37
GLP1R P43220 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
SPTLC2 O15270 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8631272 0.90 AVPR1A (0.42) AVPR2AVPR1AHSD11B1CHRM1ABCB11
Hydrochloric Acid SCHEMBL8630833 0.89 AVPR2 (0.41) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8629715 0.88 AVPR1A (0.43) AVPR2AVPR1APPARGHSD11B1CHRM1
Hydrochloric Acid SCHEMBL8628394 0.88 AVPR2 (0.43) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8630315 0.88 AVPR1A (0.45) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8634655 0.88 HSD11B1 (0.45) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8627439 0.86 AVPR1A (0.41) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8634126 0.86 AVPR2 (0.41) AVPR2AVPR1AHSD11B1CHRM1ABCB11
SCHEMBL8627201 0.83 AVPR1A (0.46) AVPR2AVPR1APOLBHSD11B1SMO
SCHEMBL8628513 0.81 AVPR1A (0.44) AVPR2AVPR1AHSD11B1CHRM1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed