SCHEMBL8632634

SCHEMBL8632634

ONC1c2ccccccc3ccccc3c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
WDR5 P61964 1/20 0.37
CYP1A2 P05177 3/20 0.37
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2A6 P11509 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HIF1A Q16665 1/20 0.37
EPHX1 P07099 1/20 0.37
MMP3 P08254 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
KDM1A O60341 1/20 0.36
NR4A1 P22736 1/20 0.35
NR4A2 P43354 1/20 0.35
NR4A3 Q92570 1/20 0.35
MTNR1A P48039 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16361430 0.64 HDAC3 (0.50) TSHRHDAC8ATM
Phenanthrene SCHEMBL28634294 0.64 HSD17B10 (0.86) WDR5CYP1A2ALDH1A1TSHRHSD17B10
SCHEMBL4377802 0.64 ALDH1A1 (0.85) CYP1A2ALDH1A1TSHRHSD17B10CYP2A6
SCHEMBL5971471 0.63 CYP1A2 (0.49) KDM4EWDR5CYP1A2ALDH1A1TSHR
SCHEMBL8564442 0.63 ALDH1A1 (0.46) KDM4ECYP1A2ALDH1A1TSHRHSD17B10
Phenanthrene SCHEMBL9994190 0.61 CYP2A6 (0.92) CYP1A2ALDH1A1TSHRHSD17B10CYP2A6
Phenanthrene SCHEMBL201780 0.61 ALDH1A1 (0.92) WDR5CYP1A2ALDH1A1TSHRHSD17B10
SCHEMBL8972474 0.60 ALDH1A1 (0.48) KDM4ECYP1A2ALDH1A1TSHRHSD17B10
Phenanthrene SCHEMBL2321409 0.59 ALDH1A1 (0.86) WDR5CYP1A2ALDH1A1TSHRHSD17B10
Phenanthrene SCHEMBL30702393 0.58 ALDH1A1 (0.71) KDM4EWDR5CYP1A2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850234-A1 NOVEL HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF PAIN AND USE THEREOF BIOCHEM PHARMA INC (CA) 1998-07-01 EP claimed
WO-1997003978-A1 NOVEL HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF PAIN AND USE THEREOF BIOCHEM PHARMA INC. (CA) 1997-02-06 WO claimed