SCHEMBL8633259

SCHEMBL8633259

NS(=O)(=O)c1ccccc1-c1n[nH]cc1-c1ccccn1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.40
CA1 P00915 4/20 0.40
IDO1 P14902 2/20 0.38
EDNRA P25101 1/20 0.38
CA9 Q16790 3/20 0.37
ALOX5AP P20292 2/20 0.37
FEN1 P39748 2/20 0.37
MAPK1 P28482 1/20 0.37
CA12 O43570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967288 0.82 EDNRA (0.49) CA2CA1EDNRACA9ALOX5AP
SCHEMBL1667127 0.82 EDNRA (0.49) CA2CA1EDNRACA9ALOX5AP
SCHEMBL7778063 0.81 CA2 (0.51) CA2CA1CA9CA12
SCHEMBL8632289 0.80 AKR1B1 (0.40) CA2CA1CA9CA12
SCHEMBL8630958 0.80 LRRK2 (0.48) CA2CA1IDO1
SCHEMBL8697589 0.79 ALOX5AP (0.47) CA2CA1EDNRACA9ALOX5AP
SCHEMBL8627632 0.78 CA1 (0.42) CA2CA1CA9CA12
SCHEMBL8634777 0.78 CA1 (0.40) CA2CA1CA9CA12
SCHEMBL8629397 0.78 ALOX5AP (0.40) CA2CA1CA9ALOX5APFEN1
SCHEMBL3463943 0.77 KDM4E (0.48) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed