SCHEMBL8633838

SCHEMBL8633838

C=CCC1CN(c2ccncc2)CCN1c1ccc(O)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.34
MAPT P10636 5/20 0.33
ALDH1A1 P00352 3/20 0.33
GAA P10253 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
KDM4E B2RXH2 3/20 0.33
DRD4 P21917 2/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
PKM P14618 1/20 0.33
MEN1 O00255 1/20 0.32
GFER P55789 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8699660 0.82 GAA (0.37) CHKAMAPTALDH1A1GAANPSR1
Hydrochloric Acid SCHEMBL8634754 0.75 GSK3B (0.45) CHKAMAPTALDH1A1GAATDP1
SCHEMBL7399577 0.73 CHKA (0.43) CHKAMAPTALDH1A1GAATDP1
SCHEMBL7334978 0.72 CHKA (0.61) CHKAMAPTALDH1A1GAATDP1
SCHEMBL8778789 0.66 CHKA (0.48) CHKADRD2DRD3ADRB2NCF1
SCHEMBL10883096 0.65 CHKA (0.46) CHKAALDH1A1KDM4EDRD2DRD3
SCHEMBL7335333 0.63 GABRA1 (0.47) CHKAMAPTALDH1A1GAATDP1
SCHEMBL8565666 0.62 MAPT (0.40) CHKAMAPTALDH1A1GAATDP1
SCHEMBL28956405 0.62 TDP1 (0.40) MAPTALDH1A1GAATDP1LMNA
SCHEMBL27930045 0.61 MAPT (0.53) CHKAMAPTGAANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed