SCHEMBL8634103

SCHEMBL8634103

C=CCN(C)CCC1(C)CCCc2cc(F)ccc2N1C(=O)c1ccc(NC(=O)c2ccccc2Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 11/20 0.41
AVPR2 P30518 8/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
NR1I2 O75469 1/20 0.40
RORA P35398 1/20 0.40
RORC P51449 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
RORB Q92753 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
AVPR1B P47901 1/20 0.38
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8634039 0.76 LMNA (0.45) AVPR1AAVPR2LMNATP53AVPR1B
Hydrochloric Acid SCHEMBL8661682 0.76 LMNA (0.44) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL8634101 0.76 NR1I2 (0.40) AVPR1AAVPR2LMNATP53NR1I2
SCHEMBL8652482 0.73 AVPR1A (0.42) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL8627357 0.73 AVPR2 (0.42) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL8634013 0.73 AVPR1A (0.42) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL8632578 0.72 AVPR2 (0.44) AVPR1AAVPR2LMNATP53AVPR1B
Hydrochloric Acid SCHEMBL8632582 0.70 AVPR2 (0.46) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL4687985 0.69 AVPR2 (0.51) AVPR1AAVPR2LMNATP53AVPR1B
SCHEMBL8651882 0.68 AVPR2 (0.44) AVPR1AAVPR2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed