SCHEMBL8634113

SCHEMBL8634113

Nc1nc(N)c2c(n1)CC/C(=N/OCc1cccc(C(F)(F)F)c1)C2

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAOB P27338 4/20 0.40
DHFR P00374 1/20 0.38
APP P05067 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634117 1.00 IDO1 (0.44) IDO1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8633331 0.84 MGMT (0.40) CYP2D6DHFR
SCHEMBL8630922 0.74 IDO1 (0.45) IDO1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8990302 0.74 EGFR (0.39) MAOB
SCHEMBL8990299 0.74 EGFR (0.39) MAOB
SCHEMBL4377734 0.70 IDO1 (0.50) IDO1MAOB
SCHEMBL8633053 0.70 HTR2C (0.37) MAOB
Hydrochloric Acid SCHEMBL4388271 0.69 IDO1 (0.51) IDO1MAOB
SCHEMBL4384916 0.66 MAOB (0.46) IDO1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4410979 0.65 MEN1 (0.48) IDO1CYP2C19MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712281-A Insecticidal substituted-2,4-diamino-5,6,7,8-tetrahydroquinazolines FMC CORPORATION (US) 1998-01-27 US disclosed
US-5536725-A Insecticidal substituted-2,4-diamino-5,6,7,8-tetrahydroquinazolines FMC CORPORATION (US) 1996-07-16 US disclosed